Gestrinone is not entirely an anabolic steroid and it didn’t start out that way too. The drug was brought into the marker as a contraceptive. However, after going through the chemical trails, it couldn’t live up to what it was required for. During the 80s, the drug was known to come with androgenic properties and later some estrogenic, progestational, anti-progestational and anti-estrogenic properties were found. Gestrinone was then modified into ‘tetrahydrogestrinone’ (THG). Both the terms are used to signify it.
How is Gestrinone used for bodybuilding?
Even now, the drug is not commonly known to fulfill anabolic requirements. It is used for treating endometriosis. The oral drug helps inhibit gonadotropins that are released by our pituitary gland. This androgen and progesterone receptor ligand is not ideal for bodybuilding, but it is not like you cannot use it either. The structure of THG comes into the notice of fitness freaks. TGH is related to Gestrinone and has potential to work like a proper steroid. However, when compared to other steroids, Trenbolone gets more preference than this.
For people who take steroids don’t usually consider the fact that the strong steroids like Trenbolone are only suggested for animal use. They are banned for human use, but many still take the risks of using it. The dangers of designer steroids are obvious, especially when the users don’t know what ingredients have been used, what the unexpected side effects are, and more.
Many bodybuilders and athletes believe that THG can be bought over the counter, but that’s not true. THG is often considered to be Trenbolone and Gestrinone, as these two are often in comparison.
Mechanism of Action for Gestrinone
Before you consider using Gestrinone, you ought to know that THG has not gone through much of studies and research, and people don’t know much about its advantages and disadvantages. People who look to buy steroids promote anabolic potential, but there is an amount of reduced androgenic properties. The drug is responsible for developing the secondary sex male characteristics, but it converts the testosterone into estrogen, and the process is called aromatization.
Men can face effects like having breast tissues or gynecomastia. Potential of water retention, bloating, and increased fat, are common too. Women can face virilization, and that means having masculine effects in their body.
It is safe to use Gestrinone?
Before using any form of anabolic steroids it is essential to know the side effects or the adverse reactions of the drug. You should not consider the benefits of the drug. The same goes for Gestrinone implants, injections and pills. Any other drug that can mimic the effects of this drug must also be taken under consideration. The risk increases when users tend to stack THG with more compounds like HGH, testosterone, and other dosages. The drug does help us have better size and strength gain, but the side effects are quite harmful too. This is an androgen and progesterone receptor ligand, but that can have both negative and positive impacts on our body.